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Cat. No. Product Name Target Signaling Pathways
T7831 Nitecapone

Others; Transferase Metabolism; Others
Nitecapone 是一个具有口服活性的、短效的儿茶酚-O-甲基转移酶(COMT)的抑制剂。它具有胃肠道保护和抗氧化活性,能够清除活性氧和一氧化氮,防止脂质过氧化。
T38823 sulfo-DGN462 sodium

sulfo-DGN462 sodium

Sulfo-DGN462 sodium undergoes degradation to DGN462 when subjected to culture medium and plasma. DGN462, a highly effective DNA-alkylating agent, exhibits anti-tumor properties that are particularly active against acute myeloid leukemia (AML).
T79873 TNG-462

Histone Methyltransferase Chromatin/Epigenetic
TNG-462(化合物1143)作为一种口服有效的PRMT5抑制剂,适用于研究MTAP缺失型及/或MTA累积型癌症。
T81060 Sulfo-SPDB-DGN462

Sulfo-SPDB-DGN462为一种ADC活性连接剂,毒素DGN462通过可裂解的Sulfo-SPDB linker偶联形成。DGN462是一种DNA烷基化剂,对抗肿瘤(如急性髓系白血病[AML])表现出有效性。
T35881 Resolvin E2

Resolvin E2 (RvE2) is a member of the specialized pro-resolving mediator (SPM) family of bioactive lipids.1It is produced from eicosapentaenoic acidviaan 18-HEPE intermediate, which is formed by aspirin-acetylated COX-2-mediated oxidation of EPA, by 5-lipoxygenase (5-LO) in human polymorphonuclear (PMN) neutrophils.2,3RvE2 (20 ng/animal) inhibits increases in inflammatory exudate neutrophil infiltration in a mouse model of peritonitis induced by zymosan A .3Hepatic RvE2 levels are increased in m...

化合物

Nitecapone
Cat.No: T7831
Synonym:
Target: Others, Transferase
sulfo-DGN462 sodium
Cat.No: T38823
Synonym: sulfo-DGN462 sodium
Target:
TNG-462
Cat.No: T79873
Synonym:
Target: Histone Methyltransferase
Sulfo-SPDB-DGN462
Cat.No: T81060
Synonym:
Target:
Resolvin E2
Cat.No: T35881
Synonym:
Target:
TargetMol Loading
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