Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T7831 |
Nitecapone
|
Others; Transferase | Metabolism; Others |
Nitecapone 是一个具有口服活性的、短效的儿茶酚-O-甲基转移酶(COMT)的抑制剂。它具有胃肠道保护和抗氧化活性,能够清除活性氧和一氧化氮,防止脂质过氧化。 | |||
T38823 |
sulfo-DGN462 sodium
sulfo-DGN462 sodium |
||
Sulfo-DGN462 sodium undergoes degradation to DGN462 when subjected to culture medium and plasma. DGN462, a highly effective DNA-alkylating agent, exhibits anti-tumor properties that are particularly active against acute myeloid leukemia (AML). | |||
T79873 |
TNG-462
|
Histone Methyltransferase | Chromatin/Epigenetic |
TNG-462(化合物1143)作为一种口服有效的PRMT5抑制剂,适用于研究MTAP缺失型及/或MTA累积型癌症。 | |||
T81060 | Sulfo-SPDB-DGN462 | ||
Sulfo-SPDB-DGN462为一种ADC活性连接剂,毒素DGN462通过可裂解的Sulfo-SPDB linker偶联形成。DGN462是一种DNA烷基化剂,对抗肿瘤(如急性髓系白血病[AML])表现出有效性。 | |||
T35881 |
Resolvin E2
|
||
Resolvin E2 (RvE2) is a member of the specialized pro-resolving mediator (SPM) family of bioactive lipids.1It is produced from eicosapentaenoic acidviaan 18-HEPE intermediate, which is formed by aspirin-acetylated COX-2-mediated oxidation of EPA, by 5-lipoxygenase (5-LO) in human polymorphonuclear (PMN) neutrophils.2,3RvE2 (20 ng/animal) inhibits increases in inflammatory exudate neutrophil infiltration in a mouse model of peritonitis induced by zymosan A .3Hepatic RvE2 levels are increased in m... |